PerkinElmer

Receptor Ligand Binding

OF

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 653 Products and Services

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LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

The EZ Reader instrument is available outside the EU. Please contact your local representative for further information.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.
PerkinElmer

Protein A PVT 500 MG

Protein A-coated SPA beads, for capturing antibodies in proximity-based radiometric scintillation assays.
List Price : 760.00 EUR

Thyroxine, ([125I]-T4), L-[125I]-, 250µCi (9.25MBq), Specific Activity: 135-165µCi (5.00-6.11MBq)/µg

NEX111 L-3,5-Diiodothyronine is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1196.00 EUR
Receptor-expressing cell lines

ValiScreen Histamine H1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

YSI PDE 25X2G

SPA (scintillation proximity assay) beads designed for the capture of [3H]AMP or [3H]GMP on specially prepared yttrium silicate beads.
List Price : 30200.00 EUR
List Price : 3621.00 EUR
PerkinElmer

Glutathione PVT 25X2G

Glutathione-coated SPA beads, for capturing GST-tagged proteins in proximity-based radiometric scintillation assays.
List Price : 50600.00 EUR
PerkinElmer

Membrane Target Systems: Calcitonin AM2 (ADM) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 823.00 EUR

2`-Deoxycytidine-5`-triphosphate, 5-[125I]iodo-, Tetraammonium Salt, 100µCi (3.7MBq)

Deoxycytidine triphosphate (dCTP) is a nucleoside triphosphate that is used whenever DNA is synthesized, such as in the polymerase chain reaction. 125I dCTP may be used to produce cDNA transcripts of viral or mRNA.
List Price : 1350.00 EUR
PerkinElmer

ProfilerPro Kinase Peptide Substrate 32, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 32 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 544.00 EUR

α-Bungarotoxin, [125I]-Tyr54-, High Specific Activity, 50 µCi

α-bungarotoxin extracted from venom of the Taiwanese banded krait (Bungarus multicinctus) binds the nicotinic acetylcholine receptor found at the neuromuscular junction and the 7 nicotinic acetylcholine receptor in the brain.
List Price : 793.00 EUR

SCH 23390, [N-Methyl-3H]

SCH-23390 (halobenzazepine), tritiated on the N-methyl group. SCH-23390 acts as an antagonist at the dopamine D1 receptor.
Price Range : 732.00 EUR - 4003.00 EUR

ANGIOTENSIN I (human), [125I]Tyr4-, 10µCi (370kBq), Species Activity:2200Ci (81.4TBq/mmol)

NEX101 Angiotensin, a protein, causes blood vessels to constrict, and drives blood pressure up. It is part of the renin-angiotensin system, which is a major target for drugs that lower blood pressure. Angiotensin also stimulates the release of aldosterone from the adrenal cortex.
List Price : 1056.00 EUR
PerkinElmer

Membrane Target Systems: Adenosine A2a (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Adenosine A2a (human) receptor, in HEK-293 cells.
List Price : 823.00 EUR
Receptor-expressing cell lines

ValiScreen Vasopressin V1b (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

WAY100635, [METHOXY-3H], 250 uCi

WAY-100635, tritiated on the methoxy group. WAY-100635 acts as an antagonist at serotonin 5-HT1A receptors. It also acts as an agonist at dopamine D4 receptors.
List Price : 5100.00 EUR
Receptor-expressing cell lines

ValiScreen N-formyl Peptide (FPRL1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Anti-sheep YSI 500 MG

Anti-sheep-coated SPA beads, for capturing sheep IgG antibodies in proximity-based radiometric scintillation assays.
List Price : 760.00 EUR
PerkinElmer

Streptavidin YSI 250MG YTTRIUM

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 2483.00 EUR
PerkinElmer

Membrane Target Systems: Neuropeptide NPFF1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuropeptide NPFF1 receptor, in CHO-K1 cells.
List Price : 823.00 EUR
PerkinElmer

ProfilerPro Kinase Peptide Substrate 13, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 13 for kinase assays (inhibiton, target discovery, lead optimization)
List Price : 665.00 EUR

Chloramphenicol, [Ring-3,5-3H]

Chloramphenicol, tritiated at the ring-3,5 position. Chloramphenicol is a broad spectrum antibiotic that binds to a receptor site on the 50S subunit of the bacterial ribosome, inhibiting peptidyl transferase.
Price Range : 2652.00 EUR - 5800.00 EUR

MIP-1α (human, recombinant), [125I], 5µCi

NEX298 [125I]-MIP-1α is useful in RIA, receptor studies and crosslinking experiments in the research into immune regulation.
List Price : 905.00 EUR
PerkinElmer

CHO cell membranes, 10 mg

Wild Type Subtype CHO-K1 (chinese hamster) Control Membrane 10mg frozen suspension cell membrane. Shipped on dry ice.
List Price : 490.00 EUR

Enkephalin, [Tyrosyl-2,6-3H(N)]- (2-D-Penicillamine, 5-D-Penicillamine) (DPDPE)

2-D-Penicillamine, 5-D-Penicillamine (DPDPE), tritiated on the tyrosyl group. Cyclic peptide, sequence: Tyr-D-Pen-Gly-Phe-D-Pen-OH. DPDPE is a synthetic enkephalin opioid peptide that acts as an agonist at delta opiate receptors (δ-opioid receptor, DOR).
Price Range : 1366.00 EUR - 6600.00 EUR

IP-10 (human, recombinant), [125I]-, Bolton-Hunter Labeled, 25µCi

NEX348 IP-10 acts at the CXCR3 receptor and attracts T cells, particularly activated T cells.
List Price : 2222.00 EUR

RX 821002, [6,7-3H(N)]-

RX 821002, tritiated at the 6,7 position. RX 821002 acts as an antagonist at α2-adrenoceptors.
List Price : 2882.00 EUR
Receptor-expressing cell lines

ValiScreen Serotonin 5HT-1A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

UniFilter-96 GF/B, White 96-well Barex Microplate with GF/B filter of 1 µm poresize

GF/B glassfibre filter-bottom 96-well microplate, for receptor binding assays using a vacuum manifold.
List Price : 982.00 EUR
Receptor-expressing cell lines

ValiScreen Glucagon - R (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Streptavidin YSI 75MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 760.00 EUR
PerkinElmer

Membrane Target Systems: Epidermal Growth Factor Receptor EGF membrane preparation

Cell membranes prepared from A431 cells containing human endogenous EGF receptor.
List Price : 823.00 EUR
PerkinElmer

Dopamine Transporter (human) Cell Line

Our stable recombinant cell lines express a variety of receptors for binding and functional assays.
List Price : 15600.00 EUR
Receptor-expressing cell lines

ValiScreen Prostanoid DP (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
Receptor-expressing cell lines

ValiScreen Neuropeptide FF NPFF2s (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Vasopressin V2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human Vasopressin V2 receptor, 400 units.
List Price : 823.00 EUR
PerkinElmer

Membrane Target Systems: Neurotensin NTS1(Leu194) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human neurotensin NTS1 (Leu194) receptor, 400 units.
List Price : 800.00 EUR

Astemizole, [O-Methyl-3H]

Astemizole (Hismanal) tritiated at the O-methyl group. Atemizole is an antagonist of the histamine H1-receptor and has been shown to block hERG potassium channels.
Price Range : 986.00 EUR - 9800.00 EUR
PerkinElmer

Membrane Target Systems: Ghrelin (human) membrane preparation, inCHO-K1 cells. 400 Units

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 726.00 EUR

"Receptor Ligand Binding" 1-50 of 653 Products and Services

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