PerkinElmer

Receptor Ligand Binding

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Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

 

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"Receptor Ligand Binding" 1-50 of 763 Products and Services

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LabChip EZ Reader

EZ READER, SHIP LEVEL

The EZ Reader can help to save time and money in your laboratory by identifying the most promising lead candidates faster.

MICROBETA FILTERMAT-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use.

UNIFILTER-96 CELL HARVESTER SS

Speed and simplicity are the primary strengths of the Unifilter Harvester.

MICROBETA FILTERMAT-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the FilterMate Harvester. From beginning to end, the FilterMate system is easy to use. Need additional information? Click on the tabs in the product details section below.

OMNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the OmniFilter Harvester.

UNIFILTER-24 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

UNIFILTER-96 CELL HARVESTER

Speed and simplicity are the primary strengths of the Unifilter Harvester.

(+)-Pentazocine, [Ring-1,3-3H]-, 25µCi (925kBq)

25 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 833.00 EUR

Ketanserin Hydrochloride (R41 468), [Ethylene-3H]-, 250µCi (9.25MBq)

250 µCi quantities of tritiated Ketanserin hydrochloride are available for your research.
List Price : 2735.00 EUR

WAY100635, [METHOXY-3H], 250 uCi

250 µCi quantities of [METHOXY-3H]-WAY100635 are available for your research.
List Price : 3936.00 EUR

(+)-Pentazocine, [Ring-1,3-3H]-,250µCi (9.25MBq)

250 µCi quantities of [Ring-1, 3-3H]-(+)-Pentazocine are available for your research.
List Price : 2710.00 EUR

Paroxetine, [Phenyl-6`-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Phenyl-6'-3H]-Paroxetine are available for your research.
List Price : 2990.00 EUR
PerkinElmer

Membrane Target Systems: Dopamine D44 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Dopamine D44 (human) receptor, in CHO-K1 cells.
List Price : 784.00 EUR

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 50µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 2479.00 EUR
PerkinElmer

Membrane Target Systems: Melanocortin MC5 (mouse) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 784.00 EUR
PerkinElmer

HDAC (Histone Deacylase) Substrate A, for LabChip EZ Reader

Fluorescently-labelled Substrate A peptide (Acetylated) for Epigenetic Assays (Enzyme inhibiton, target discovery, lead optimization)
List Price : 544.00 EUR

AB-MECA, [125I]-(4-Amino-3-[125I]iodobenzyl-5`-N-)-, 10µCi

AB-MECA is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method and is purified by reversed phase HPLC.
List Price : 1395.00 EUR

Interleukin-1β (human, recombinant), [125I], 25µCi

NEX232 Interleukin-1 (IL-1) refers to a group of three polypeptides (interleukin-1 alpha (IL-1α), interleukin-1 beta (IL-1β) and interleukin-1 receptor antagonist (IL-1Ra)), that play a central role in the regulation of immune and inflammatory responses.

IL-1β is a pro-inflammatory cytokine involved in immune defense against infection.

List Price : 2746.00 EUR

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 250µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 5600.00 EUR

CGP 39653, [Propyl-2,3,3H]-, 1mCi (37MBq)

1 mCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 6400.00 EUR

[125I]Tyr0-Corticotropin Releasing Factor (ovine), 10 µCi

NEX217 Corticotropin-releasing hormone (CRH), originally named corticotropin-releasing factor (CRF), and also called corticoliberin, is a polypeptide hormone and neurotransmitter involved in the stress response.
List Price : 1404.00 EUR
PerkinElmer

Membrane Target Systems: N-formyl Peptide (FPRL1) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 784.00 EUR
PerkinElmer

HDAC (Histone Deacylase) Substrate B, for LabChip EZ Reader

Fluorescently-labelled Substrate A peptide (Acetylated) for Epigenetic Assays (Enzyme inhibiton, target discovery, lead optimization)
List Price : 529.00 EUR

ANGIOTENSIN I (human), [125I]Tyr4-, 10µCi (370kBq), Species Activity:2200Ci (81.4TBq/mmol)

NEX101 Angiotensin, a protein, causes blood vessels to constrict, and drives blood pressure up. It is part of the renin-angiotensin system, which is a major target for drugs that lower blood pressure. Angiotensin also stimulates the release of aldosterone from the adrenal cortex.
List Price : 1005.00 EUR

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Ring, Methylenes-3H(N)]-Histamine Dihydrochloride are available for your research.
List Price : 1169.00 EUR

Norepinephrine, Levo-[7-3H]-, 5mCi (185MBq)

5 mCi quantities of Levo-[7-3H]-Norepinephrine are available for your research.
List Price : 10700.00 EUR

Interleukin-1β (human, recombinant), [125I], 10µCi

NEX232 Interleukin-1 (IL-1) refers to a group of three polypeptides (interleukin-1 alpha (IL-1α), interleukin-1 beta (IL-1β) and interleukin-1 receptor antagonist (IL-1Ra)), that play a central role in the regulation of immune and inflammatory responses.

IL-1β is a pro-inflammatory cytokine involved in immune defense against infection.

List Price : 2028.00 EUR
PerkinElmer

Streptavidin PVT 50MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
List Price : 238.00 EUR

Substance-P (9-Sar, 11-Met(O2)), [2-Prolyl-3,4-3H]-, 50µCi (1.85MBq)

50 µCi quantities of tritiated Substance-P are available for your research.
List Price : 2944.00 EUR

8-Hydroxy-DPAT, [Propyl-2,3-ring-1,2,3-3H]-, 250µCi (9.25MBq)

250 µCi quantities of [Propyl-2, 3-ring-1, 2, 3-3H]-8-Hydroxy-DPAT are available for your research.
List Price : 1608.00 EUR

Lysergic Acid Diethylamide, 2-[125I]iodo-(+), 10µCi

NEX199 Preparations have been shown to be active in binding to the serotonin receptors. LSD affects a large number of the G protein coupled receptors, including all dopamine receptor subtypes, and all adrenoreceptor subtypes, as well as many others. LSD binds to most serotonin receptor subtypes except for 5-HT3 and 5-HT4.
List Price : 1032.00 EUR

Hydroxytryptamine Creatinine Sulfate (Serotonin), 5-[1,2-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of 5-[1, 2-3H(N)]-Hydroxytryptamine Creatinine Sulfate (Serotonin) are available for your research.
List Price : 999.00 EUR
Receptor-expressing cell lines

ValiScreen Adrenergic beta 2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

CGP 39653, [Propyl-2,3,3H]-, 25µCi (925kBq)

25 µCi quantities of [Propyl-2, 3, 3H]-CGP 39653 are available for your research
List Price : 781.00 EUR
PerkinElmer

Membrane Target Systems: Neuromedin U NMU1 (human) membrane preparation

Cell membranes prepared from cells stably-transfected with human Neuromedin U NMU1 receptor, in HEK-293 cells.
List Price : 784.00 EUR
PerkinElmer

Membrane Target Systems: Serotonin 5HT-5A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
List Price : 784.00 EUR

Vasopressin (Linear), V-1A Antagonist (Phenylacetyl1, 0-Me-D-Tyr2, [125I-Arg6]-),50µCi

NEX310 [125I]-Phenylacetyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr-NH2 is useful in receptor studies and autoradiography for the localization and characterization of Vasopressin V1A receptors.
List Price : 2509.00 EUR

Ketanserin Hydrochloride (R41 468), [Ethylene-3H]-, 25µCi (925kBq)

25 µCi quantities of tritiated Ketanserin hydrochloride are available for your research.
List Price : 823.00 EUR

Bradykinin, [2,3-Prolyl-3,4-3H(N)]-, 50µCi (1.85MBq)

50 µCi quantities of [2, 3-Prolyl-3, 4-3H(N)]-Bradykinin are available for your research.
List Price : 2063.00 EUR

CGRP (human), [125I]-, 50µCi

NEX354 Human CGRP binds to human CGRP receptors in the central nervous system and peripheral nervous system. [125I]-CGRP (human) will be useful in the characterization of CGRP receptors.
List Price : 2265.00 EUR
List Price : 2610.00 EUR
PerkinElmer

WGA PS Imaging Beads 50 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based scintillation assays.
List Price : 44.00 EUR
PerkinElmer

Membrane Target Systems: Transporter Dopamine (human) membrane preparation

Cell membranes prepared from cells stably-transfected with Transporter Dopamine receptor, in CHO-K1 cells.
List Price : 784.00 EUR

AF-DX 384, [2,3-Dipropylamino-3H]-, 250µCi (9.25MBq)

250 µCi quantities of AF-DX 384, [2, 3-Dipropylamino-3H]- are available for your research.
List Price : 2607.00 EUR

RTI-55, [125I]-, 25µCi (925kBq)

NEX272 [125I]-RTI-55 is an excellent radioligand for the study of the dopamine transporter sites using either tissue homogenates or autoradiographic methods--especially in regions of low receptor density.
List Price : 1060.00 EUR

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]-, 1mCi (37MBq)

1 mCi quantities of [Ring, Methylenes-3H(N)]-Histamine Dihydrochloride are available for your research.
List Price : 2542.00 EUR

Goat anti-rabbit IgG, [125I], 100µCi (3.7MBq)

Affinity purified goat anti-rabbit IgG is radioiodinated with no carrier added 125I using a modification of the Hunter and Greenwood method1 and is purified by gel filtration chromatography. This method predominantly labels tyrosine residues.
List Price : 939.00 EUR
Receptor-expressing cell lines

ValiScreen Melanocortin MC1 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

CGS 21680, [Carboxyethyl-3H(N)]-, 250µCi (9.25MBq)

250 µCi quantities of [Carboxyethyl-3H(N)]-CGS 21680 are available for your research.
List Price : 2454.00 EUR

"Receptor Ligand Binding" 1-50 of 763 Products and Services

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